IMR OpenIR

浏览/检索结果: 共18条,第1-10条 帮助

已选(0)清除 条数/页:   排序方式:
Design, Synthesis, Biological Activity and Molecular Docking Study of Coumarin Derivatives Bearing 2-Methylbiphenyl Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2019, 卷号: 35, 期号: 3, 页码: 410-417
作者:  Ma Junjie;  Huang Kun;  Ni Xin;  Chen Roufen;  Xu Boxuan;  Wang Cuifang
收藏  |  浏览/下载:112/0  |  提交时间:2021/02/02
GROWTH  POTENT  Coumarin  2-Methylbiphenyl  Anticancer activity  PD-1/PD-L1 inhibitory activity  Molecular docking  
Design, Synthesis and Biological Activities of N-(Furan-2-ylmethyl)-1H-indole-3-carboxamide Derivatives as Epidemal Growth Factor Receptor Inhibitors and Anticancer Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 3, 页码: 365-372
作者:  Zhang Lan;  Deng Xinshan;  Wu Jiaofeng;  Meng Guangpeng;  Liu Congchong;  Chen Guzhou;  Zhao Qingchun;  Hu Chun
收藏  |  浏览/下载:151/0  |  提交时间:2021/02/02
MOLECULAR TARGETED DRUGS  TYROSINE KINASE  CANCER-CELLS  EGFR  RESISTANCE  POTENT  DISCOVERY  NSCLC  Anticancer activity  Epidemal growth factor receptor(EGFR) inhibitor  N-( Furan-2-ylmethyl)-1H-indole3-carboxamide derivative  
Design, Synthesis and Biological Activities of N-(Furan-2-ylmethyl)-1H-indole-3-carboxamide Derivatives as Epidemal Growth Factor Receptor Inhibitors and Anticancer Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 3, 页码: 365-372
作者:  Zhang Lan;  Deng Xinshan;  Wu Jiaofeng;  Meng Guangpeng;  Liu Congchong;  Chen Guzhou;  Zhao Qingchun;  Hu Chun
收藏  |  浏览/下载:146/0  |  提交时间:2021/02/02
MOLECULAR TARGETED DRUGS  TYROSINE KINASE  CANCER-CELLS  EGFR  RESISTANCE  POTENT  DISCOVERY  NSCLC  Anticancer activity  Epidemal growth factor receptor(EGFR) inhibitor  N-( Furan-2-ylmethyl)-1H-indole3-carboxamide derivative  
Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:  Ma Junjie;  Hu Gang;  Xie Lijun;  Chen Lei;  Xu Boxuan;  Gong Ping
收藏  |  浏览/下载:126/0  |  提交时间:2021/02/02
POTENT  INHIBITORS  ONCRASIN-1  DISCOVERY  Benzothiazole  Semicarbazone  Antitumor activity  
Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:  Ma Junjie;  Hu Gang;  Xie Lijun;  Chen Lei;  Xu Boxuan;  Gong Ping
收藏  |  浏览/下载:145/0  |  提交时间:2021/02/02
POTENT  INHIBITORS  ONCRASIN-1  DISCOVERY  Benzothiazole  Semicarbazone  Antitumor activity  
Design, Synthesis and Antitumor Activity of Novel 6,7-Dimethoxyquinazoline Derivatives Containing Diaryl Urea Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 766-773
作者:  Hou Yunlei;  Wu Shasha;  Ma Longsheng;  Bai Jinying;  Liu Zijian;  Zhao Yanfang
收藏  |  浏览/下载:123/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASES  BIOLOGICAL EVALUATION  HIGHLY POTENT  INHIBITOR  IDENTIFICATION  GROWTH  DISCOVERY  SORAFENIB  EGFR  6,7-Dimethoxyquinazoline derivative  Diaryl urea scaffold  Cytotoxic activity  
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:  Sun ChiYu;  Li YangSheng;  Shi AiLong;  Li YaFei;  Cao RuiFang;  Ding HuaiWei;  Yin QingQing;  Zhang LiJuan;  Zheng HuaChuan;  Song HongRui
收藏  |  浏览/下载:153/0  |  提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY  BASAL-CELL CARCINOMA  INHIBITORS  DISCOVERY  DESIGN  ANTAGONISTS  IDENTIFICATION  VISMODEGIB  CANCER  POTENT  Aryl cycloaliphatic amine  Antiproliferative activity  Hedgehog signaling  
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:  Sun ChiYu;  Li YangSheng;  Shi AiLong;  Li YaFei;  Cao RuiFang;  Ding HuaiWei;  Yin QingQing;  Zhang LiJuan;  Zheng HuaChuan;  Song HongRui
收藏  |  浏览/下载:142/0  |  提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY  BASAL-CELL CARCINOMA  INHIBITORS  DISCOVERY  DESIGN  ANTAGONISTS  IDENTIFICATION  VISMODEGIB  CANCER  POTENT  Aryl cycloaliphatic amine  Antiproliferative activity  Hedgehog signaling  
Synthesis and Antitumor Activities of Novel 4-Morpholinothieno3,2-dpyrimidine Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 1, 页码: 75-81
作者:  Song Kaizhen;  Ma Junjie;  Wang Xiao;  Gong Ping;  Zhao Yanfang
收藏  |  浏览/下载:84/0  |  提交时间:2021/02/02
CANCER  POTENT  INHIBITOR  KINASE  2-Hydrazinyl-4-morpholinothieno3,2-dpyrimidine  Antitumor activity  Cytotoxic activity  
Pharmacophore-based design, synthesis, and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-substituted benzyl)amino) propanamides as cholesteryl ester transfer protein (CETP) inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2014, 卷号: 25, 期号: 2, 页码: 299-304
作者:  Zhao DongMei;  Li WenYan;  Shi YuFang;  Xiong XuQiong;  Song Shuai;  Hao ChenZhou;  Cheng MaoSheng;  Shen JingKang
收藏  |  浏览/下载:163/0  |  提交时间:2021/02/02
CHIRAL N,N-DISUBSTITUTED TRIFLUORO-3-AMINO-2-PROPANOLS  POTENT INHIBITORS  DISCOVERY  TRANSPORT  Cholesteryl ester transfer protein  CETP inhibitors  Pharmacophore  Virtual screening  Synthesis